Peptide Handbook
Hormonal & Immune Peptides

Thymosin Alpha-1

Immune Modulator — TLR2/TLR9 Agonist

Updated April 14, 2026

What is Thymosin Alpha-1?

A 28-amino-acid peptide originally isolated from thymic tissue (thymosin fraction 5) by Allan Goldstein in 1977. Thymosin alpha-1 (Tα1) is a bidirectional immune modulator — it upregulates immune response in immunodeficiency while dampening excessive inflammation in sepsis and autoimmunity. Activates dendritic cells via TLR2 and TLR9, enhances NK cell cytotoxicity, and promotes T-cell maturation. Approved in over 35 countries (trade name Zadaxin) for hepatitis B and as an immune adjuvant.

Research Profile

Structure 28 amino acids (~3,108 Da) — N-acetylated
Targets TLR2/TLR9, dendritic cells, NK cells, T-cell maturation
Research Focus Immune modulation, viral hepatitis, vaccine adjuvancy, sepsis, cancer immunotherapy
Reconstitution Bacteriostatic water — 1.6 mg/mL
Stability 21 days at 2–8°C
Key distinction: Bidirectional immune modulator — uniquely capable of both upregulating suppressed immunity and dampening hyperinflammation. Approved in 35+ countries with decades of clinical safety data.

Published Research

[1] Goldstein AL et al. Thymosin alpha1: isolation and sequence analysis of an immunologically active thymic polypeptide. Proc Natl Acad Sci USA 1977;74:725-729 — PubMed 265542
[2] Romani L et al. Thymosin alpha1 activates dendritic cell tryptophan catabolism and establishes a regulatory environment for balance of inflammation and tolerance. Blood 2006;108:2265-2274 — PubMed 16740584
Research Use Only. All products sold by Lumen Peppers are intended solely for in vitro research and laboratory purposes. They are not drugs, supplements, or foods. Nothing on this page constitutes medical advice. Researchers are responsible for compliance with all applicable regulations. Last updated: April 14, 2026.

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